3
Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T12128 | Mutant IDH1-IN-2 | Isocitrate Dehydrogenase (IDH) | |
Mutant IDH1-IN-2 is a mutant Isocitrate dehydrogenase (IDH) proteins inhibitor | |||
T11611 | IDH1 Inhibitor 2 | Dehydrogenase | |
IDH1 Inhibitor 2 (compound 13) is a potent IDH1 inhibitor via direct covalent modification of His315 (IC50: 110 nM). | |||
T7307 | Vorasidenib | PVM/MA,AG-881 | Isocitrate Dehydrogenase (IDH) |
Vorasidenib (PVM/MA) is an inhibitor of mutant isocitrate dehydrogenase (IDH; IC50s = 31.9 and 31.7 nM for IDH1R132H and IDH2R140Q, respectively) |